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Found 708 from Kafrelsheikh University
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM50520843(CHEMBL4585732)
Affinity DataKi:  1.30nMAssay Description:Inhibition of recombinant human carbonic anhydrase 12 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM50456991(CHEMBL2237247)
Affinity DataKi:  1.80nMAssay Description:Inhibition of human cytosolic carbonic anhydrase 2 by stopped-flow CO2 hydrase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM50569044(CHEMBL4872457)
Affinity DataKi:  1.80nMAssay Description:Inhibition of human CA9 by stopped- flow CO2 hydration assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 7(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM10880(AZA | AZA2 | AZM acetazolamide | Acerazolamide, AA...)
Affinity DataKi:  2.5nMAssay Description:Inhibition of human recombinant carbonic anhydrase 7 incubated for 15 mins prior to testing by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM50457006(CHEMBL4211148)
Affinity DataKi:  2.60nMAssay Description:Inhibition of human cytosolic carbonic anhydrase 2 by stopped-flow CO2 hydrase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM50582974(CHEMBL5082587)
Affinity DataKi:  3.30nMAssay Description:Inhibition of human CA12 preincubated for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM50520838(CHEMBL4579656)
Affinity DataKi:  3.60nMAssay Description:Inhibition of recombinant human carbonic anhydrase 12 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 4(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM50230939(CHEMBL4067135)
Affinity DataKi:  4nMAssay Description:Inhibition of human recombinant carbonic anhydrase 4 incubated for 15 mins prior to testing by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM50582963(CHEMBL5075785)
Affinity DataKi:  4.20nMAssay Description:Inhibition of human CA12 preincubated for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM50567601(CHEMBL4857595)
Affinity DataKi:  4.30nMAssay Description:Inhibition of recombinant human CA9 pre-incubated for 15 mins measured by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM50334354(4-(3-(4-fluorophenyl)ureido)benzenesulfonamide | 4...)
Affinity DataKi:  4.5nMAssay Description:Inhibition of recombinant human CA12 pre-incubated for 15 mins measured by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM50334354(4-(3-(4-fluorophenyl)ureido)benzenesulfonamide | 4...)
Affinity DataKi:  4.5nMAssay Description:Inhibition of human CA12 measured after 15 mins by stopped flow carbon dioxide anhydrase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM50334354(4-(3-(4-fluorophenyl)ureido)benzenesulfonamide | 4...)
Affinity DataKi:  4.5nMAssay Description:Inhibition of human CA12 preincubated for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM50334354(4-(3-(4-fluorophenyl)ureido)benzenesulfonamide | 4...)
Affinity DataKi:  4.5nMAssay Description:Inhibition of human carbonic anhydrase 12 assessed as inhibition constant incubated for 15 mins prior to testing by phenol red based stopped-flow CO2...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM50456991(CHEMBL2237247)
Affinity DataKi:  4.5nMAssay Description:Inhibition of human transmembrane carbonic anhydrase 9 by stopped-flow CO2 hydrase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM50334354(4-(3-(4-fluorophenyl)ureido)benzenesulfonamide | 4...)
Affinity DataKi:  4.5nMAssay Description:Inhibition of recombinant human carbonic anhydrase 12 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM50520834(CHEMBL4533369)
Affinity DataKi:  4.70nMAssay Description:Inhibition of recombinant human carbonic anhydrase 9 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM50569035(CHEMBL4867387)
Affinity DataKi:  4.80nMAssay Description:Inhibition of human CA2 by stopped- flow CO2 hydration assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM50591870(CHEMBL5203094)
Affinity DataKi:  5.10nMAssay Description:Inhibition of human carbonic anhydrase 2 assessed as inhibition constant incubated for 15 mins prior to testing by phenol red based stopped-flow CO2 ...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM50567598(CHEMBL4853209)
Affinity DataKi:  5.10nMAssay Description:Inhibition of recombinant human CA12 pre-incubated for 15 mins measured by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM50591870(CHEMBL5203094)
Affinity DataKi:  5.20nMAssay Description:Inhibition of human carbonic anhydrase 12 assessed as inhibition constant incubated for 15 mins prior to testing by phenol red based stopped-flow CO2...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM50513674(CHEMBL4458485)
Affinity DataKi:  5.20nMAssay Description:Inhibition of recombinant human carbonic anhydrase 9 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM50569040(CHEMBL4873532)
Affinity DataKi:  5.5nMAssay Description:Inhibition of human CA9 by stopped- flow CO2 hydration assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM10880(AZA | AZA2 | AZM acetazolamide | Acerazolamide, AA...)
Affinity DataKi:  5.60nMAssay Description:Inhibition of human CA12 preincubated for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM10880(AZA | AZA2 | AZM acetazolamide | Acerazolamide, AA...)
Affinity DataKi:  5.60nMAssay Description:Inhibition of recombinant human carbonic anhydrase 12 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM10880(AZA | AZA2 | AZM acetazolamide | Acerazolamide, AA...)
Affinity DataKi:  5.70nMAssay Description:Inhibition of recombinant human CA12 pre-incubated for 15 mins measured by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM10880(AZA | AZA2 | AZM acetazolamide | Acerazolamide, AA...)
Affinity DataKi:  5.70nMAssay Description:Inhibition of human CA12 by stopped- flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM10880(AZA | AZA2 | AZM acetazolamide | Acerazolamide, AA...)
Affinity DataKi:  5.70nMAssay Description:Inhibition of human carbonic anhydrase 12 assessed as inhibition constant incubated for 15 mins prior to testing by phenol red based stopped-flow CO2...More data for this Ligand-Target Pair
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM10880(AZA | AZA2 | AZM acetazolamide | Acerazolamide, AA...)
Affinity DataKi:  5.70nMAssay Description:Inhibition of human CA12 measured after 15 mins by stopped flow carbon dioxide anhydrase assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM50567599(CHEMBL4847847)
Affinity DataKi:  5.90nMAssay Description:Inhibition of recombinant human CA2 pre-incubated for 15 mins measured by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM50230950(CHEMBL4096684)
Affinity DataKi:  5.90nMAssay Description:Inhibition of human recombinant carbonic anhydrase 2 incubated for 15 mins prior to testing by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM10880(AZA | AZA2 | AZM acetazolamide | Acerazolamide, AA...)
Affinity DataKi:  6nMAssay Description:Inhibition of recombinant human carbonic anhydrase 12 preincubated with enzyme for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM50582959(CHEMBL5087786)
Affinity DataKi:  6.20nMAssay Description:Inhibition of human CA9 preincubated for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM50513674(CHEMBL4458485)
Affinity DataKi:  6.30nMAssay Description:Inhibition of recombinant human carbonic anhydrase 12 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM50567598(CHEMBL4853209)
Affinity DataKi:  6.5nMAssay Description:Inhibition of recombinant human CA9 pre-incubated for 15 mins measured by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM50230942(CHEMBL4085952)
Affinity DataKi:  6.60nMAssay Description:Inhibition of human recombinant carbonic anhydrase 2 incubated for 15 mins prior to testing by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM50230940(CHEMBL4069845)
Affinity DataKi:  6.80nMAssay Description:Inhibition of human recombinant carbonic anhydrase 2 incubated for 15 mins prior to testing by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM50569041(CHEMBL4864064)
Affinity DataKi:  7.10nMAssay Description:Inhibition of human CA9 by stopped- flow CO2 hydration assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM50456997(CHEMBL4213947)
Affinity DataKi:  7.10nMAssay Description:Inhibition of human cytosolic carbonic anhydrase 2 by stopped-flow CO2 hydrase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM50582971(CHEMBL5074754)
Affinity DataKi:  7.30nMAssay Description:Inhibition of human CA12 preincubated for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM50567598(CHEMBL4853209)
Affinity DataKi:  7.40nMAssay Description:Inhibition of recombinant human CA2 pre-incubated for 15 mins measured by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM50591866(CHEMBL5203184)
Affinity DataKi:  7.5nMAssay Description:Inhibition of human carbonic anhydrase 12 assessed as inhibition constant incubated for 15 mins prior to testing by phenol red based stopped-flow CO2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM50569035(CHEMBL4867387)
Affinity DataKi:  7.60nMAssay Description:Inhibition of human CA9 by stopped- flow CO2 hydration assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM50230937(CHEMBL4095939)
Affinity DataKi:  7.70nMAssay Description:Inhibition of human recombinant carbonic anhydrase 2 incubated for 15 mins prior to testing by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM50520842(CHEMBL4547434)
Affinity DataKi:  7.70nMAssay Description:Inhibition of recombinant human carbonic anhydrase 12 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM50520829(CHEMBL4536441)
Affinity DataKi:  7.80nMAssay Description:Inhibition of recombinant human carbonic anhydrase 12 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM50567599(CHEMBL4847847)
Affinity DataKi:  7.90nMAssay Description:Inhibition of recombinant human CA12 pre-incubated for 15 mins measured by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM50569044(CHEMBL4872457)
Affinity DataKi:  8nMAssay Description:Inhibition of human CA2 by stopped- flow CO2 hydration assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM50582974(CHEMBL5082587)
Affinity DataKi:  8.10nMAssay Description:Inhibition of human CA9 preincubated for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM50569039(CHEMBL4860334)
Affinity DataKi:  8.10nMAssay Description:Inhibition of human CA12 by stopped- flow CO2 hydration assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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